Anesthetic (local); antiarrhythmic (class IB). Long-acting, membrane stabilizing agent against ventricular arrhythmia. Originally developed as a local anesthetic.
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参考文献
• Groningsson, K., et al.: Anal. Profiles Drug Subs., 14, 207 (1971)
• Kronberg, G.H., et al.: J. Med. Chem., 16, 739 (1971)
• Davies, P.S., et al.: Drugs, 64, 937 (1971)
• Duce, R., et al.: J. Pharmacol. Exp. Ther., 179, 580 (1971)